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Human microdosing for the prediction of patient response

Paul T. Henderson, C. Pan

Bioanalysis March 1, 2010 DOI: 10.4155/bio.10.3 (opens in new tab)

Study at a glance

AI-extracted from the abstract
Characteristics Review Peer reviewed
Topics Microdosing
Key findings Argues that microdosing, originally developed in molecular toxicology, is now being applied to medical diagnostics, with recent efforts focusing on prognostic and predictive diagnostics to improve disease detection and treatment.

Abstract

Microdosing allows study of the behavior of drugs via the administration of doses so low they are unlikely to produce whole-body effects, but of sufficient concentration to allow the determination of absorption, distribution, metabolism and excretion (ADME). Microdosing was recently reviewed elsewhere [1,2]; although most effort to date has focused on pharmacokinetic (PK) predictions to accelerate drug development, microdosing was born out of molecular toxicology research [3-10] and is now extending to medical diagnostics applications. Here, we provide a brief overview of microdosing for drug development, followed by a description of recent efforts to implement prognostic and predictive diagnostics aimed at improving detection and treatment of human disease.