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Acute LSD effects on response inhibition neural networks

André Schmidt, Felix Müller, Claudia Lenz, Patrick C. Dolder, Yasmin Schmid, Davide Zanchi, Undine E. Lang, Matthias E. Liechti, Stefan Borgwardt

Psychological Medicine October 2, 2017 DOI: 10.1017/s0033291717002914 (opens in new tab)

Study at a glance

AI-extracted from the abstract
Characteristics Randomized controlled trial Placebo-controlled Double-blind Peer reviewed
Sample size 18
Population Healthy subjects
Intervention LSD
Dose 100 µg
Topics LSD
Keywords Visual hallucination Parahippocampal gyrus Cingulate cortex Prefrontal cortex Visual cortex Postcentral gyrus Placebo Audiology Cognition
Citations 62
Key findings LSD-induced activation of the serotonin 2A receptor impairs response inhibition by disrupting hippocampal-prefrontal cortex networks, and this disruption is linked to visual hallucinations.

Abstract

Abstract Background Recent evidence shows that the serotonin 2A receptor (5-hydroxytryptamine2A receptor, 5-HT 2A R) is critically involved in the formation of visual hallucinations and cognitive impairments in lysergic acid diethylamide (LSD)-induced states and neuropsychiatric diseases. However, the interaction between 5-HT 2A R activation, cognitive impairments and visual hallucinations is still poorly understood. This study explored the effect of 5-HT 2A R activation on response inhibition neural networks in healthy subjects by using LSD and further tested whether brain activation during response inhibition under LSD exposure was related to LSD-induced visual hallucinations.

Methods: In a double-blind, randomized, placebo-controlled, cross-over study, LSD (100 µg) and placebo were administered to 18 healthy subjects. Response inhibition was assessed using a functional magnetic resonance imaging Go/No-Go task. LSD-induced visual hallucinations were measured using the 5 Dimensions of Altered States of Consciousness (5D-ASC) questionnaire.

Results: Relative to placebo, LSD administration impaired inhibitory performance and reduced brain activation in the right middle temporal gyrus, superior/middle/inferior frontal gyrus and anterior cingulate cortex and in the left superior frontal and postcentral gyrus and cerebellum. Parahippocampal activation during response inhibition was differently related to inhibitory performance after placebo and LSD administration. Finally, activation in the left superior frontal gyrus under LSD exposure was negatively related to LSD-induced cognitive impairments and visual imagery.

Conclusion: Our findings show that 5-HT 2A R activation by LSD leads to a hippocampal–prefrontal cortex-mediated breakdown of inhibitory processing, which might subsequently promote the formation of LSD-induced visual imageries. These findings help to better understand the neuropsychopharmacological mechanisms of visual hallucinations in LSD-induced states and neuropsychiatric disorders.

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