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Prefrontal cortical distribution of muscarinic M2 and cannabinoid-1 (CB1) receptors in adult male mice with or without chronic adolescent exposure to Δ9-tetrahydrocannabinol.

Miguel Garzón, June Chan, Ken Mackie, Virginia M Pickel

Cerebral cortex (New York, N.Y. : 1991) November 21, 2022 DOI: 10.1093/cercor/bhac024 (opens in new tab)

Study at a glance

AI-extracted from the abstract
Characteristics Experimental animal study Peer reviewed
Population Adult C57BL/6 J male mice that received vehicle or escalating-dose Δ9-THC during adolescence
Dose escalating dose
Measures electron microscopic dual CB1R and M2R immunolabeling, M2R-immunogold density
Topics Cannabis
Keywords Cannabinoid Cholinergic Prelimbic Ultrastructure
Key findings Adolescent Δ9-THC treatment increased plasmalemmal M2R-immunogold density specifically in large dendrites receiving input from CB1R-labeled terminals and decreased cytoplasmic M2R-immunogold density in small spines of the prelimbic prefrontal cortex. The authors conclude that Δ9-THC engagement of CB1Rs during adolescence increases M2R surface accumulation in large proximal dendrites and decreases M2R cytoplasmic expression in small spines.

Abstract

Chronic adolescent administration of marijuana's major psychoactive compound, ∆9-tetrahydrocannabinol (Δ9-THC), produces adaptive changes in adult social and cognitive functions sustained by prelimbic prefrontal cortex (PL-PFC). Memory and learning processes in PL-PFC neurons can be regulated through cholinergic muscarinic-2 receptors (M2R) and modulated by activation of cannabinoid-1 receptors (CB1Rs) targeted by Δ9-THC. Thus, chronic exposure to Δ9-THC during adolescence may alter the expression and/or distribution of M2Rs in PL-PFC neurons receiving CB1R terminals. We tested this hypothesis by using electron microscopic dual CB1R and M2R immunolabeling in adult C57BL/6 J male mice that had received vehicle or escalating dose of Δ9-THC through adolescence. In vehicle controls, CB1R immunolabeling was mainly localized to axonal profiles virtually devoid of M2R but often apposing M2R-immunoreactive dendrites and dendritic spines. The dendrites received inputs from CB1R-labeled or unlabeled terminals, whereas spines received asymmetric synapses exclusively from axon terminals lacking CB1Rs. Adolescent Δ9-THC significantly increased plasmalemmal M2R-immunogold density exclusively in large dendrites receiving input from CB1R-labeled terminals. In contrast, cytoplasmic M2R-immunogold density decreased in small spines of the Δ9-THC-treated adult mice. We conclude that Δ9-THC engagement of CB1Rs during adolescence increases M2R plasmalemmal accumulation in large proximal dendrites and decreases M2R cytoplasmic expression in small spines of PL-PFC.

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