Amphetamine derivatives interact with both plasma membrane and secretory vesicle biogenic amine transporters.
Molecular Pharmacology December 1, 1993 S Schuldiner, S Steiner-Mordoch, R Yelin et al.
The interaction of fenfluramine, 3,4-methylenedioxymethamphetamine (MDMA), and p-chloroamphetamine (PCA) with the platelet plasma membrane serotonin transporter and the vesicular amine transporter were studied using both transport and binding measurements. Fenfluramine is apparently a substrate for the plasma membrane transporter, and consequently inhibits both serotonin transport and...
DOI: 10.1016/s0026-895x(25)13357-9 (opens in new tab)
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Serotonin
Chromaffin granules
Blood platelets
Cell membrane
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